YM-58790 1 Ligand-Linker Conjugates 1 H2O/c1-25(5-3-4-6-25)7-10-8-31-17-13(16(27)24(17)14(10)18(28)29)22-15(26)12(23-30-2)11-9-32-19(20)21-11

H2O/c1-25(5-3-4-6-25)7-10-8-31-17-13(16(27)24(17)14(10)18(28)29)22-15(26)12(23-30-2)11-9-32-19(20)21-11

Chemical Name: methyl 4-hydroxybenzoate

while Proglumide does not influence the basal amylase release at concentrations between 0-3 mM

Mice LD50 values are 215

4 μM one hour after oral administration and undetectable levels 23 hours after administration

YM-58790 1 Ligand-Linker Conjugates 1 H2O/c1-25(5-3-4-6-25)7-10-8-31-17-13(16(27)24(17)14(10)18(28)29)22-15(26)12(23-30-2)11-9-32-19(20)21-11YM 58790 is a potent antagonist of M3 muscarinic receptor, with Ki of 15 nM. Product information CAS Number: 214558 72 2 Molecular Weight: 466. 01 Formula: C27H32ClN3O2 Chemical Name: 1 {[4 (methylamino)phenyl]methyl}piperidin 4 yl N (diphenylmethyl)carbamate hydrochloride Smiles: Cl. CNC1=CC=C(CN2CCC(CC2)OC(=O)NC(C2=CC=CC=C2)C2=CC=CC=C2)C=C1 InChiKey: WKHYQXVQUGLLOZ UHFFFAOYSA N InChi: InChI=1S C27H31N3O2. ClH c1 28 24 14 12 21(13 15 24)20 30 18 16